SCHEMBL8051980

SCHEMBL8051980

c1cnc(CCc2ccncn2)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
HSP90AA1 P07900 1/20 0.37
HRH1 P35367 2/20 0.36
HRH3 Q9Y5N1 2/20 0.36
HRH4 Q9H3N8 1/20 0.36
RPS6KA5 O75582 1/20 0.35
KCNH3 Q9ULD8 1/20 0.34
CYP1B1 Q16678 1/20 0.33
SORD Q00796 1/20 0.33
P2RX7 Q99572 1/20 0.32
LMNA P02545 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
PDE10A Q9Y233 1/20 0.32
FLT1 P17948 1/20 0.32
KDR P35968 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23685443 0.83 HRH1 (0.55) CYP1A2CYP2D6HRH1HRH3HRH4
SCHEMBL30746342 0.78 KCNH2 (0.50) CYP1A2CYP2D6TAAR1
SCHEMBL1514838 0.78 KCNH2 (0.50) CYP1A2CYP2D6TAAR1
SCHEMBL11361045 0.74
SCHEMBL1661146 0.74
SCHEMBL2015773 0.74
SCHEMBL1666852 0.74
SCHEMBL9573114 0.74
SCHEMBL16399930 0.74
SCHEMBL11361047 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948792-A POTENT AND SELECTIVE ANTAGONISTS FOR MUSCARINIC M.SUB.3 RECEPTORS WITH LITTLE SIDE EFFECTS. BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-09-07 US claimed
EP-0930298-A1 FLUORINATED 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-07-21 EP claimed
US-10669371-B2 Benzothienothiophene isoindigo polymers BASF SE (DE) 2020-06-02 US disclosed
US-6040449-A USEFUL FOR FORMING FLUORINE CONTAINING 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES, USEFUL AS ANTAGONIST FOR MUSCARINIC M3 RECEPTORS AND LESS SIDE EFFECT BANYU PHARMACEUTICAL CO LTD (JP) 2000-03-21 US disclosed
US-5948792-A POTENT AND SELECTIVE ANTAGONISTS FOR MUSCARINIC M.SUB.3 RECEPTORS WITH LITTLE SIDE EFFECTS. BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-09-07 US disclosed