SCHEMBL8055784

SCHEMBL8055784

CCN(SC)C1CCN(CCC(C)(C(=O)OC)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 4/20 0.49
TACR2 P21452 3/20 0.49
TACR1 P25103 3/20 0.49
KCNH2 Q12809 2/20 0.41
CACNA1I Q9P0X4 1/20 0.41
CCR5 P51681 2/20 0.39
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
OPRM1 P35372 2/20 0.36
OPRL1 P41146 1/20 0.36
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 2/20 0.35
USP2 O75604 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042308 0.90 TACR2 (0.51) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL8032648 0.89 TACR3 (0.53) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL296855 0.84 TACR3 (0.49) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL296221 0.84 TACR3 (0.68) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL370294 0.84 TACR3 (0.48) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL296394 0.82 TACR3 (0.50) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL296889 0.82 TACR3 (0.52) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL371169 0.81 TACR3 (0.51) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL296888 0.79 TACR3 (0.45) TACR3TACR2TACR1KCNH2CACNA1I
SCHEMBL297581 0.78 TACR3 (0.45) TACR3TACR2TACR1KCNH2CACNA1I

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009033995-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-03-19 WO disclosed