SCHEMBL8058044

SCHEMBL8058044

C#Cc1ccc(O)c(C(=O)OCC)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.64
CA1 P00915 4/20 0.64
CA2 P00918 4/20 0.64
CA7 P43166 4/20 0.64
CA9 Q16790 4/20 0.64
CA14 Q9ULX7 4/20 0.64
KMT2A Q03164 2/20 0.50
EGFR P00533 2/20 0.48
TSHR P16473 2/20 0.47
HSD17B2 P37059 1/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
HSP90AA1 P07900 1/20 0.43
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5485097 0.87 TSHR (0.55) CA12CA1CA2CA7CA9
SCHEMBL18094303 0.83 TSHR (0.46) CA12CA1CA2CA7CA9
SCHEMBL7711875 0.82 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL5736404 0.81 CA12 (0.47) CA12CA1CA2CA7CA9
SCHEMBL1641611 0.78 CA12 (0.74) CA12CA1CA2CA7CA9
SCHEMBL39259 0.78 CA12 (1.00) CA12CA1CA2CA7CA9
SCHEMBL29457603 0.78 CA12 (1.00) CA12CA1CA2CA7CA9
SCHEMBL8028947 0.78 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL27415591 0.77 TSHR (0.41) CA12CA1CA2CA7CA9
SCHEMBL10570974 0.77 CA12 (0.74) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0613468-B1 Substituted salicylic acids for the treatment of autoimmune diseases PHARMACIA & UPJOHN AB (SE) 2000-07-12 EP disclosed
CN-1042631-C Novel substituted salicylic acids KABI PHARMACIA AB (SE) 1999-03-24 CN disclosed
US-5556855-A TREATMENT OF AUTOIMMUNE DISEASES PHARMACIA AB (SE) 1996-09-17 US disclosed
US-5403930-A Chemical intermediate for drugs used in autoimmune diseases PHARMACIA AB (SE) 1995-04-04 US disclosed
EP-0613468-A1 NOVEL SUBSTITUTED SALICYCLIC ACIDS Pharmacia & Upjohn Aktiebolag (SE) 1994-09-07 EP disclosed
CN-1088918-A The salicylic acid compounds of new replacement KABI PHARMACIA AB (SE) 1994-07-06 CN disclosed
US-5302718-A Used for treating autoimmune diseases KABI PHARMACIA AB (SE) 1994-04-12 US disclosed
WO-1993010094-A1 NOVEL SUBSTITUTED SALICYCLIC ACIDS KABI PHARMACIA AB (SE) 1993-05-27 WO disclosed