SCHEMBL8059115

SCHEMBL8059115

COC(=O)c1cc2nc[nH]c2c(F)c1Nc1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.40
CYP3A4 P08684 2/20 0.38
P2RY6 Q15077 1/20 0.38
P2RY14 Q15391 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NR4A2 P43354 1/20 0.38
TTBK1 Q5TCY1 1/20 0.37
TTBK2 Q6IQ55 1/20 0.37
TSHR P16473 1/20 0.37
HTT P42858 1/20 0.37
QPCT Q16769 2/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
CYP3A5 P20815 1/20 0.35
CSF1R P07333 1/20 0.35
SLC6A3 Q01959 1/20 0.34
EGFR P00533 2/20 0.34
KDR P35968 2/20 0.34
ERBB2 P04626 1/20 0.34
CDK1 P06493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4545994 0.89 MAPT (0.43) MKNK1TSHRCSF1RKDM4ENPC1
SCHEMBL1038046 0.85 MAPT (0.42) L3MBTL1NR4A2TSHRHTTEGFR
SCHEMBL8059139 0.84 MAP2K1 (0.43) L3MBTL1NR4A2TSHRHTTCSF1R
SCHEMBL30746852 0.82 NR4A2 (0.40) MKNK1CYP3A4P2RY6P2RY14L3MBTL1
SCHEMBL1038083 0.82 NR4A2 (0.40) MKNK1CYP3A4P2RY6P2RY14L3MBTL1
SCHEMBL1078430 0.79 CYP2C9 (0.45) CYP3A4NR4A2CSF1RKDM4ENPC1
SCHEMBL19119163 0.78 NR4A2 (0.36) CYP3A4P2RY6P2RY14L3MBTL1NR4A2
SCHEMBL3886544 0.77 MEN1 (0.45) KMT2ASMN1; SMN2
SCHEMBL1075382 0.74 MAP2K1 (0.43) CYP3A4EGFRKDM4EKMT2ASMN1; SMN2
SCHEMBL1077717 0.73 NR4A2 (0.40) MKNK1CYP3A4P2RY6P2RY14NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009036020-A1 MEK INHIBITORS CONTAINING A ZINC BINDING MOIETY CURIS, INC. (US) 2009-03-19 WO disclosed