SCHEMBL805927

SCHEMBL805927

OCCc1cc(NCCN2CCOCC2)cc(-c2ccc(Oc3ccc(F)cc3)cc2)n1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 14/20 0.73
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
PDE5A O76074 1/20 0.46
KCNH2 Q12809 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL805910 0.84 SCN9A (1.00) SCN9ANPC1RAB9A
SCHEMBL787531 0.83 SCN9A (1.00) SCN9A
SCHEMBL29421433 0.83 SCN9A (1.00) SCN9A
SCHEMBL21236966 0.76 SCN9A (0.53) SCN9A
SCHEMBL16174381 0.75 SCN9A (0.66) SCN9ATSHR
SCHEMBL17076600 0.74 SCN9A (0.57) SCN9ANPC1RAB9AKDM4EALDH1A1
SCHEMBL14920033 0.73 SCN9A (0.83) SCN9AKCNH2KDM4EALDH1A1HPGD
SCHEMBL787277 0.71 SCN9A (1.00) SCN9A
SCHEMBL787278 0.71 SCN9A (0.86) SCN9A
SCHEMBL21236944 0.70 SCN9A (0.77) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616441-B1 PYRIDINE COMPOUNDS AND THE USES THEREOF PURDUE PHARMA LP (US) 2019-08-07 EP disclosed
WO-2012035421-A2 PYRIDINE COMPOUNDS AND THE USES THEREOF PURDUE PHARMA L.P. (US) 2012-03-22 WO disclosed