SCHEMBL8060641

SCHEMBL8060641

CNC1CS(=O)(=O)c2cc(C(=O)N=C(N)N)ccc21

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 4/20 0.42
ADRA1D P25100 1/20 0.42
HTR2A P28223 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SLC9A2 Q9UBY0 1/20 0.42
HTR2B P41595 3/20 0.41
HTR7 P34969 2/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056274 0.83 HTR2B (0.46) HTR2BHTR7
SCHEMBL8060754 0.82 HTR2B (0.41) SLC9A1HTR2BHTR7
SCHEMBL8045374 0.82 HTR2B (0.46) HTR2BHTR7
SCHEMBL8045075 0.82 HTR2B (0.48) HTR2BHTR7
SCHEMBL8063051 0.81
SCHEMBL8045040 0.81 HTR2B (0.44) HTR2BHTR7
SCHEMBL8062798 0.80 SLC6A2 (0.46) SLC6A3
SCHEMBL8060820 0.80 HTR2B (0.41) HTR2BHTR7
SCHEMBL8057135 0.78 HTR2B (0.41) SLC9A1HTR2BHTR7CYP3A4CYP2C9
SCHEMBL8060778 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed