SCHEMBL8060645

SCHEMBL8060645

N#CC(O)C(Cc1ccccc1)NC(=O)Cn1c(-c2ccc(F)cc2)ncc(NC(=O)OCc2ccccc2)c1=O

nearest known ligand 0.67

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6558412 0.89 ELANE (0.73) ELANE
SCHEMBL8064266 0.85 ELANE (0.71) ELANE
SCHEMBL8061828 0.85 ELANE (0.63) ELANE
SCHEMBL6556185 0.85 ELANE (0.69) ELANE
SCHEMBL6556195 0.85 ELANE (0.69) ELANE
SCHEMBL6556190 0.85 ELANE (0.69) ELANE
SCHEMBL8060598 0.84 ELANE (0.70) ELANE
SCHEMBL6558392 0.84 ELANE (0.71) ELANE
SCHEMBL6558258 0.84 ELANE (0.79) ELANE
SCHEMBL8059711 0.84 ELANE (0.61) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080738-A USEFUL AS CHYMASE INHIBITORS AND CAN BE USED FOR THE PROPHYLAXIS AND TREATMENT OF VARIOUS DISEASES CAUSED BY CHYMASE, SUCH AS THOSE CAUSED BY ANGIOTENSIN II YOSHITOMI PHARMACEUTICALS INDUSTRIES, LTD. (JP) 2000-06-27 US disclosed
EP-0940400-A1 NOVEL HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USES THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-08 EP disclosed