SCHEMBL8064828

SCHEMBL8064828

O=C(/C=C/c1cc[n+]([O-])cc1)Nc1cccc(-c2cccc(-n3c(=O)c(Cc4cccnc4)nc4cccnc43)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.42
BTK Q06187 3/20 0.42
ITK Q08881 2/20 0.42
NAMPT P43490 5/20 0.38
HDAC4 P56524 3/20 0.37
MEF2D Q14814 3/20 0.37
DHFR P00374 2/20 0.37
SIRT2 Q8IXJ6 2/20 0.37
SIRT1 Q96EB6 2/20 0.37
SIRT3 Q9NTG7 2/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
POLB P06746 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
FLT3 P36888 2/20 0.35
BLK P51451 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7493481 1.00 EGFR (0.42) EGFRBTKITKNAMPTHDAC4
SCHEMBL6794724 0.92 EGFR (0.44) EGFRBTKITKNAMPTHDAC4
SCHEMBL6794732 0.92 EGFR (0.44) EGFRBTKITKNAMPTHDAC4
Hydrochloric Acid SCHEMBL6796140 0.92 EGFR (0.47) EGFRBTKITKNAMPTHDAC4
Hydrochloric Acid SCHEMBL6796145 0.92 EGFR (0.47) EGFRBTKITKNAMPTHDAC4
SCHEMBL6797628 0.91 EGFR (0.45) EGFRBTKITKNAMPTHDAC4
SCHEMBL6797634 0.91 EGFR (0.45) EGFRBTKITKNAMPTHDAC4
SCHEMBL7360146 0.90 EGFR (0.43) EGFRBTKITKNAMPTHDAC4
SCHEMBL7360140 0.90 EGFR (0.43) EGFRBTKITKNAMPTHDAC4
SCHEMBL8063774 0.89 EGFR (0.40) EGFRBTKITKNAMPTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117875-A Pyrido (2,3-B) pyrazine derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-12 US disclosed