SCHEMBL806501

SCHEMBL806501

COc1cc2c(cc1OC)[C@@]1(C)CC[C@H](I)C(C)(C)C1CC2

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
POLA1 P09884 11/20 0.48
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
CYP3A4 P08684 1/20 0.40
SOD1 P00441 1/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15978371 1.00 POLA1 (0.48) POLA1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL15978302 0.91 POLA1 (0.46) POLA1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL806502 0.82 POLA1 (0.63) POLA1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL15978299 0.82 POLA1 (0.63) POLA1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL15980588 0.77 POLA1 (0.41) POLA1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL806818 0.77 POLA1 (0.41) POLA1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL9880751 0.75 POLA1 (0.51) POLA1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL806727 0.74 SRD5A1 (0.46) NR1H2NR1H3
SCHEMBL15978295 0.74 SRD5A1 (0.46) NR1H2NR1H3
SCHEMBL15978421 0.70 POLA1 (0.34) POLA1CYP2C9TSHRCYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037069-A2 UNIQUE HALOGEN-INDUCED CYCLIZATIONS, REAGENTS THEREFOR, AND COMPOUNDS PRODUCED THEREBY THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2012-03-22 WO disclosed