SCHEMBL8065833

SCHEMBL8065833

COC(=O)/C=C/c1cncc(C=Cc2cccc(-n3c(=O)c(Cc4cccnc4)nc4cccnc43)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
EGFR P00533 2/20 0.40
BTK Q06187 2/20 0.40
ITK Q08881 1/20 0.40
NQO1 P15559 1/20 0.39
PSD A5PKW4 1/20 0.38
MAPT P10636 2/20 0.36
HKDC1 Q2TB90 2/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
PDE4B Q07343 3/20 0.36
PDE4D Q08499 1/20 0.36
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
ALDH1A1 P00352 4/20 0.35
RAD1 O60671 1/20 0.35
CFTR P13569 1/20 0.35
APEX1 P27695 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8065829 1.00 KDM4E (0.41) KDM4EKMT2ASMN1; SMN2EGFRBTK
SCHEMBL7487766 1.00 KDM4E (0.41) KDM4EKMT2ASMN1; SMN2EGFRBTK
SCHEMBL6804121 0.96 EGFR (0.43) KDM4EKMT2ASMN1; SMN2EGFRBTK
SCHEMBL6804117 0.96 EGFR (0.43) KDM4EKMT2ASMN1; SMN2EGFRBTK
SCHEMBL7490989 0.89 EGFR (0.40) KDM4EKMT2AEGFRBTKITK
SCHEMBL7490991 0.89 EGFR (0.40) KDM4EKMT2AEGFRBTKITK
SCHEMBL6798405 0.89 EGFR (0.46) KDM4EKMT2ASMN1; SMN2EGFRBTK
SCHEMBL6798410 0.89 EGFR (0.46) KDM4EKMT2ASMN1; SMN2EGFRBTK
SCHEMBL7493019 0.87 PSD (0.40) KDM4EKMT2AEGFRBTKITK
SCHEMBL8064742 0.87 PSD (0.40) KDM4EKMT2AEGFRBTKITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117875-A Pyrido (2,3-B) pyrazine derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-09-12 US disclosed