SCHEMBL8067710

SCHEMBL8067710

C/C(=N\C(C)C)N1CCc2nc(C(=O)O)sc2C1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 16/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
F10 P00742 1/20 0.36
OGA O60502 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL980083 0.80 GRM5 (0.50) GRM5NPC1RAB9AHDAC3HDAC1
SCHEMBL980081 0.80 GRM5 (0.50) GRM5NPC1RAB9AHDAC3HDAC1
SCHEMBL12035524 0.76 F10 (0.47) F10OGAHDAC3HDAC1HDAC6
SCHEMBL741699 0.75 F10 (0.46) F10OGAHDAC3HDAC1HDAC6
SCHEMBL1251008 0.74 F10 (0.50) GRM5F10
SCHEMBL741444 0.73 ADORA1 (0.55) GRM5NPC1RAB9AF10
Hydrochloric Acid SCHEMBL209036 0.73 F10 (0.49) GRM5F10
SCHEMBL207703 0.73 F10 (0.49) GRM5F10
SCHEMBL210375 0.72 ADORA1 (0.54) GRM5NPC1RAB9AF10
SCHEMBL15014912 0.70 RAD52 (0.60) GRM5NPC1RAB9AF10HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009037001-A2 NOVEL TETRAHYDROFUSEDPYRIDINES AS HISTONE DEACETYLASE INHIBITORS 4SC AG (DE) 2009-03-26 WO disclosed