SCHEMBL8068248

SCHEMBL8068248

CCOc1cc(CC)c(C(F)(F)F)cc1C(=O)Nc1cccc2c1CCN(C)C2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
KIT P10721 1/20 0.42
KCNK3 O14649 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41
RXFP1 Q9HBX9 3/20 0.41
KDR P35968 3/20 0.39
KLKB1 P03952 1/20 0.39
MAPT P10636 1/20 0.39
PTGES O14684 1/20 0.38
NR1I2 O75469 1/20 0.38
UGCG Q16739 1/20 0.38
MAP4K1 Q92918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7801341 0.92 MEN1 (0.43) MEN1KMT2AKCNK3KCNK9RXFP1
SCHEMBL8182722 0.92 KDR (0.43) MEN1KMT2AKITKDRKLKB1
SCHEMBL7799939 0.91 MEN1 (0.43) MEN1KMT2AKCNK3KCNK9RXFP1
SCHEMBL7791943 0.90 MEN1 (0.42) MEN1KMT2AKCNK3KCNK9RXFP1
SCHEMBL7792082 0.89 MEN1 (0.42) MEN1KMT2AKCNK3KCNK9RXFP1
SCHEMBL7799951 0.88 MEN1 (0.49) MEN1KMT2AMAPTNR1I2UGCG
SCHEMBL7799980 0.86 HSD17B10 (0.43) MEN1KMT2ARXFP1MAPTNR1I2
SCHEMBL7797946 0.86 KMT2A (0.43) MEN1KMT2AMAPTNR1I2UGCG
SCHEMBL7801319 0.86 KMT2A (0.43) MEN1KMT2ARXFP1MAPTNR1I2
SCHEMBL7801338 0.86 KMT2A (0.45) MEN1KMT2AMAPTNR1I2UGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025087-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-08-09 EP disclosed
WO-1999021836-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1999-05-06 WO disclosed