SCHEMBL8069310

SCHEMBL8069310

Bc1ccc([C@H]2CN([C@H](C)c3ccccc3)C(=O)CO2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.46
MAPK1 P28482 1/20 0.38
HSD11B1 P28845 2/20 0.36
GRM5 P41594 1/20 0.35
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
CYP2D6 P10635 2/20 0.34
CYP3A4 P08684 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
MDM2 Q00987 1/20 0.33
BRD4 O60885 2/20 0.33
LTA4H P09960 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2295755 0.88 KMT2A (0.46) KMT2AMAPK1HSD11B1
SCHEMBL2295888 0.88 KMT2A (0.46) KMT2AMAPK1HSD11B1
SCHEMBL2297334 0.88 KMT2A (0.46) KMT2AMAPK1HSD11B1GRM5ALDH1A1
SCHEMBL2296900 0.88 MDM2 (0.47) KMT2AMAPK1HSD11B1CYP3A4MDM2
SCHEMBL2295538 0.88 KMT2A (0.46) KMT2AMAPK1HSD11B1
SCHEMBL2298680 0.88 KMT2A (0.46) KMT2AMAPK1HSD11B1GRM5ALDH1A1
SCHEMBL2294941 0.88 MDM2 (0.47) KMT2AMAPK1HSD11B1CYP3A4MDM2
SCHEMBL2294266 0.88 MDM2 (0.47) KMT2AMAPK1HSD11B1CYP3A4MDM2
SCHEMBL917086 0.88 MDM2 (0.47) KMT2AMAPK1HSD11B1CYP3A4MDM2
SCHEMBL2296090 0.88 KMT2A (0.46) KMT2AMAPK1HSD11B1GRM5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009035159-A1 3-METHYL-2- ( (2S) -2- (4- (3-METHYL-L, 2, 4-0XADIAZ0L-5-YL) PHENYL) MORPHOLINO) -6- (PYRIMIDIN-4-YL) PYRIMIDIN-4 (3H) -ONE AS TAU PROTEIN KINASE INHIBITOR MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-19 WO disclosed