SCHEMBL8071742

SCHEMBL8071742

CCOC(=O)c1c(C(=O)c2ccc(NC(C)=O)cc2N)nnn1Cc1ccc(OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HSD17B10 Q99714 3/20 0.47
HPGD P15428 2/20 0.47
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 2/20 0.45
POLB P06746 3/20 0.45
MAPT P10636 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
ALOX15 P16050 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
RECQL P46063 1/20 0.44
AKR1C3 P42330 7/20 0.43
TSHR P16473 2/20 0.43
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8073462 0.90 MKNK2 (0.46) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL8067007 0.88 KMT2A (0.45) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL7815561 0.88 POLB (0.46) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL7827011 0.86 POLB (0.50) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL7831227 0.84 POLB (0.46) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL7829087 0.84 POLB (0.48) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL8068083 0.84 AKR1C3 (0.48) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL7828659 0.83 KDM4E (0.47) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL8073234 0.83 MEN1 (0.44) MEN1KMT2AHSD17B10HPGDALDH1A1
SCHEMBL7831536 0.81 POLB (0.44) MEN1KMT2AHSD17B10HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6093714-A AN ANTIALLERGENS FOR TREATMENT AND PREVENTION OF BRONCHIAL ASTHMA, ECZEMA, HIVES, ALLERGIC GASTROINTESTINAL TROUBLES, ALLERGIC RHINITIS, ALLERGIC CONJUNCTIVITIS MEIJI SEIKA KAISHA, LTD. (JP) 2000-07-25 US disclosed
EP-0834512-A1 TRICYCLIC BENZAZEPINE COMPOUNDS MEIJI SEIKA KAISHA LTD. (JP) 1998-04-08 EP disclosed