SCHEMBL807334

SCHEMBL807334

Nc1nc2ccccc2cc1-c1ccc(C(=O)N2CCOCC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.54
MKNK1 Q9BUB5 2/20 0.52
MKNK2 Q9HBH9 2/20 0.52
JAK2 O60674 2/20 0.52
HPGD P15428 4/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
RIPK1 Q13546 1/20 0.50
ATR Q13535 1/20 0.48
GRM2 Q14416 1/20 0.48
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ATM Q13315 1/20 0.47
JAK1 P23458 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28178640 0.74 SMN1; SMN2 (0.63) MKNK1MKNK2HPGDNPC1RIPK1
SCHEMBL8150805 0.74 HPGD (0.76) HPGDMEN1KMT2ANPC1RAB9A
SCHEMBL2227506 0.74 KCNH2 (0.77) KCNH2MKNK1
SCHEMBL807327 0.74 HPGD (0.53) HPGDNPC1RAB9AGRM2ALDH1A1
SCHEMBL13968161 0.73 KCNH2 (0.76) KCNH2JAK2
SCHEMBL2749415 0.73 KCNH2 (0.59) KCNH2MKNK1MKNK2HPGDNPC1
SCHEMBL13952297 0.72 HPGD (0.60) HPGDRIPK1ALDH1A1L3MBTL1TSHR
SCHEMBL6102102 0.72 HPGD (0.57) KCNH2MKNK1MKNK2JAK2HPGD
SCHEMBL10720943 0.71 PHGDH (0.81) HPGDKMT2AALDH1A1KDM4EL3MBTL1
SCHEMBL31428791 0.71 TSHR (0.68) HPGDNPC1RAB9AALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037108-A1 AMINOQUINOLINE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-03-22 WO disclosed