SCHEMBL8075124

SCHEMBL8075124

CC(C)(C)OC(=O)N[C@@H](Cc1cc(F)cc(F)c1)C(O)CNCc1cccc(C(F)(F)F)c1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.72
CTSD P07339 8/20 0.59
BCHE P06276 2/20 0.58
CTSB P07858 4/20 0.52
BACE2 Q9Y5Z0 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13306181 1.00 BACE1 (0.72) BACE1CTSDBCHECTSBBACE2
SCHEMBL13306696 1.00 BACE1 (0.72) BACE1CTSDBCHECTSBBACE2
SCHEMBL716159 0.92 BACE1 (0.69) BACE1CTSDBCHEBACE2
SCHEMBL715055 0.92 BACE1 (0.69) BACE1CTSDBCHEBACE2
SCHEMBL3355052 0.91 BACE1 (0.68) BACE1CTSDCTSB
SCHEMBL13306616 0.91 BACE1 (0.68) BACE1CTSDCTSB
SCHEMBL13307641 0.91 BACE1 (0.68) BACE1CTSDCTSB
SCHEMBL13334080 0.89 BACE1 (0.66) BACE1CTSDCTSBBACE2
SCHEMBL3349885 0.88 BACE1 (0.65) BACE1CTSDBCHECTSBBACE2
SCHEMBL14201296 0.88 BACE1 (0.68) BACE1CTSDCTSBBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009027601-A2 PYRAZOLE 3,5 CARBOXYLATE DERIVATIVES PREPARATION AND THERAPEUTIC APPLICATION THEREOF SANOFI-AVENTIS (FR) 2009-03-05 WO disclosed