SCHEMBL807630

SCHEMBL807630

O=C(Cc1cccc(-n2nnc3ccccc32)c1)N1CCc2[nH]nc(-c3ccncc3)c2C1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.49
CREBBP Q92793 1/20 0.49
MAPK1 P28482 7/20 0.44
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15065016 0.80 MAPK1 (0.59) BRD4CREBBPMAPK1P2RX7
SCHEMBL15082111 0.80 MAPK1 (0.59) BRD4CREBBPMAPK1P2RX7
SCHEMBL807226 0.80 MAPK1 (0.59) BRD4CREBBPMAPK1P2RX7
SCHEMBL15065457 0.78 CREBBP (0.55) BRD4CREBBPMAPK1
SCHEMBL807246 0.77 MAPK1 (0.61) BRD4CREBBPMAPK1P2RX7
SCHEMBL807232 0.77 BRD4 (0.67) BRD4CREBBPMAPK1P2RX7
SCHEMBL807192 0.77 BRD4 (0.58) BRD4CREBBPMAPK1P2RX7
SCHEMBL17868173 0.76 BRD4 (0.77) BRD4CREBBPMAPK1P2RX7
SCHEMBL807225 0.74 BRD4 (0.61) BRD4CREBBPMAPK1P2RX7
SCHEMBL807436 0.73 BRD4 (0.60) BRD4CREBBPMAPK1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012036997-A1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS SCHERING CORPORATION (US) 2012-03-22 WO disclosed