SCHEMBL8076355

SCHEMBL8076355

CCOC(=O)c1cc(C(=O)OCC)cc([N+](=O)[O-])c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.79
CA12 O43570 1/20 0.55
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA7 P43166 1/20 0.55
CA9 Q16790 1/20 0.55
CA14 Q9ULX7 1/20 0.55
MAPT P10636 4/20 0.51
KMT2A Q03164 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
ALOX5 P09917 2/20 0.50
KCNJ1 P48048 1/20 0.50
KCNH2 Q12809 1/20 0.50
RAB9A P51151 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
PKM P14618 1/20 0.49
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114367 0.96 NPC1 (0.79) NPC1CA12CA1CA2CA7
SCHEMBL584234 0.94 NPC1 (0.71) NPC1CA12CA1CA2CA7
SCHEMBL7683393 0.94 NPC1 (0.71) NPC1CA12CA1CA2CA7
SCHEMBL11170918 0.92 NPC1 (0.74) NPC1CA12CA1CA2CA7
SCHEMBL584503 0.92 NPC1 (0.69) NPC1CA12CA1CA2CA7
SCHEMBL13144461 0.92 NPC1 (0.73) NPC1CA12CA1CA2CA7
SCHEMBL5095881 0.90 NPC1 (0.71) NPC1CA12CA1CA2CA7
SCHEMBL584156 0.89 NPC1 (0.66) NPC1MAPTKMT2ASMN1; SMN2ALDH1A1
SCHEMBL91308 0.89 NPC1 (1.00) NPC1CA12CA1CA2CA7
SCHEMBL3266105 0.89 NPC1 (0.69) NPC1CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4292142-A MIXTURE OF PHTHALIC ANHYDRIDE AND MALEIC ANHYDRIDE INTERNATIONAL SYNTHETIC RUBBER CO., LTD. (GB) 1981-09-29 US claimed
CN-1314659-C Method for preparing ioxitalamic acid JIANGSU INST OF NUCLEAR MED (CN) 2007-05-09 CN disclosed
CN-1803765-A Method for preparing ioxitalamic acid JIANGSU INST OF NUCLEAR MED (CN) 2006-07-19 CN disclosed
EP-0879815-B1 Process for the preparation of the 5-nitro-isophthalic-di- C1-C4-alkyl esters BAYER AG (DE) 2000-11-02 EP disclosed
US-6002041-A Process for preparing di-C1 - C4 -alkyl 5-nitro-isophthalates BAYER AKTIENGESELLSCHAFT (DE) 1999-12-14 US disclosed
EP-0879815-A1 Process for the preparation of the 5-nitro-isophthalic-di- C1-C4-alkyl esters BAYER AG (DE) 1998-11-25 EP disclosed
WO-1993023352-A1 NITRATION SYSTEM, AND PROCESS FOR NITRATING AROMATIC COMPOUNDS NORSK HYDRO A.S (NO) 1993-11-25 WO disclosed
EP-0203957-B1 5-(3,5-DISUBSTITUTED PHENYLAZO)-2-HYDROXYBENZENE ACETIC ACIDS AND SALTS AND LACTONES THEREOF, AND PHARMACEUTICAL COMPOSITIONS OF SAID ACIDS, SALTS, AND LACTONES PHARMACIA AB (SE) 1990-03-14 EP disclosed
US-4725676-A 5-(3,5-disubstituted phenylazo)-2-hydroxybenzene-acetic acids and salts and lactones thereof having a potentially inhibitory effect on 15-hydroxy-prostaglandin dehydrogenase PHARMACIA AB (SE) 1988-02-16 US disclosed
EP-0203957-A1 5-(3,5-disubstituted phenylazo)-2-hydroxybenzene acetic acids and salts and lactones thereof, and pharmaceutical compositions of said acids, salts, and lactones. PHARMACIA AB (SE) 1986-12-10 EP disclosed
WO-1986003195-A1 NOVEL AZO COMPOUNDS PHARMACIA AB (SE) 1986-06-05 WO disclosed