SCHEMBL8077191

SCHEMBL8077191

CN1C(=O)C=C[C@@]2(C)C1CC[C@@H]1[C@H]2CC[C@]2(C)C(CNC(=O)Nc3cccc(Cl)c3Cl)CC[C@@H]12

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.56
KCNH2 Q12809 6/20 0.48
SRD5A2 P31213 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8077188 1.00 AR (0.56) ARKCNH2SRD5A2
SCHEMBL4800880 0.87 AR (0.56) ARKCNH2SRD5A2
SCHEMBL2640079 0.87 AR (0.56) ARKCNH2SRD5A2
SCHEMBL4800871 0.87 AR (0.56) ARKCNH2SRD5A2
SCHEMBL8499353 0.86 AR (0.57) ARKCNH2SRD5A2
SCHEMBL8905357 0.86 AR (0.57) ARKCNH2SRD5A2
SCHEMBL9112118 0.86 AR (0.58) ARKCNH2SRD5A2
SCHEMBL8077080 0.86 AR (0.58) ARKCNH2SRD5A2
SCHEMBL8074246 0.86 AR (0.58) ARKCNH2SRD5A2
SCHEMBL8071797 0.85 SRD5A1 (0.47) SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641208-B1 4-AZASTEROID 5-ALPHA-REDUCTASE INHIBITORS MERCK & CO INC (US) 2000-08-02 EP claimed
US-5620986-A TREATS BENIGN PROSTATIC HYPERTROPHY, SEBORRHEA, FEMALE HIRSUTISM, AND MALE AND FEMALE PATTEN BALDNESS MERCK & CO., INC. (US) 1997-04-15 US claimed
EP-0641208-A4 4-AZASTEROID 5-ALPHA-REDUCTASE INHIBITORS. MERCK & CO INC (US) 1995-08-30 EP claimed
EP-0641208-A1 4-AZASTEROID 5-ALPHA-REDUCTASE INHIBITORS MERCK & CO. INC. (US) 1995-03-08 EP claimed