SCHEMBL8077358

SCHEMBL8077358

CCOc1cc(OCC)c(C(=O)Nc2cccc3c2CCN(C(C)O)C3)cc1C(C)=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.41
CARM1 Q86X55 2/20 0.41
NR1I2 O75469 1/20 0.39
UGCG Q16739 1/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
CREBBP Q92793 2/20 0.39
TSHR P16473 2/20 0.39
CYP3A4 P08684 1/20 0.39
P2RY1 P47900 1/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
RXFP1 Q9HBX9 2/20 0.37
POLB P06746 1/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7797937 0.87 KMT2A (0.44) ACACBCARM1NR1I2UGCGKMT2A
SCHEMBL8077363 0.84 MEN1 (0.44) ACACBCARM1NR1I2UGCGKMT2A
SCHEMBL7801319 0.81 KMT2A (0.43) ACACBCARM1NR1I2UGCGKMT2A
SCHEMBL7799922 0.81 KMT2A (0.43) ACACBCARM1NR1I2UGCGKMT2A
SCHEMBL7802459 0.77 KMT2A (0.43) CARM1NR1I2UGCGKMT2AMEN1
SCHEMBL7802393 0.77 KMT2A (0.44) CARM1NR1I2UGCGKMT2AMEN1
Hydrochloric Acid SCHEMBL7791936 0.76 HSD17B10 (0.44) NR1I2UGCGKMT2AMEN1CYP3A4
Hydrochloric Acid SCHEMBL7797935 0.76 KMT2A (0.43) CARM1NR1I2UGCGKMT2AMEN1
SCHEMBL8185612 0.76 KMT2A (0.46) KMT2AMEN1TSHRCYP3A4MAPT
SCHEMBL7799938 0.76 KMT2A (0.43) ACACBCARM1NR1I2UGCGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025087-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-08-09 EP disclosed
WO-1999021836-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1999-05-06 WO disclosed