SCHEMBL8079926

SCHEMBL8079926

COc1ccc(/C=C/CCCCCC#N)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 3/20 0.44
CYP3A4 P08684 3/20 0.44
TSHR P16473 2/20 0.44
LMNA P02545 2/20 0.44
TP53 P04637 1/20 0.44
GAA P10253 1/20 0.44
LTB4R Q15722 1/20 0.44
LTB4R2 Q9NPC1 1/20 0.44
TRPA1 O75762 1/20 0.43
RELA Q04206 1/20 0.43
CYP1A2 P05177 4/20 0.42
HPGD P15428 2/20 0.42
MAPT P10636 1/20 0.42
NFKB1 P19838 1/20 0.42
APEX1 P27695 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP1A1 P04798 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8079932 1.00 KDM4E (0.44) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL28162321 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL19667752 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL15688437 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL15688436 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL17682006 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL19452377 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL2005564 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL2005561 0.82 CNR1 (0.54) KDM4EALDH1A1CYP3A4TSHRLMNA
SCHEMBL31336307 0.82 KDM4E (0.42) KDM4EALDH1A1CYP3A4TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048989-A PARASITICIDES AND ANTIBROTOZOA AGENTS WASHINGTON UNIVERSITY (US) 2000-04-11 US disclosed
US-6025511-A A MYRISTIC ACID SELECTED ANALOGS FOR INHIBITING THE BIOSYNTHESIS OF THE GLYCOSYL PHOSPHATIDYLINOSITOL (GPI) ANCHOR OF THE PARASITE WASHINGTON UNIVERSITY (US) 2000-02-15 US disclosed
US-6001869-A CONTACTING THE PARASITE WITH 2-THIENYL-UNDECENOIC ACID/10-/ WASHINGTON UNIVERSITY (US) 1999-12-14 US disclosed
US-5998642-A Thienyl-containing fatty acid glycosyl phosphatidylinosital analogues used for inhibiting parasitic activity WASHINGTON UNIVERSITY (US) 1999-12-07 US disclosed
US-5760259-A MYRISTIC ACID DERIVATIVES CAPABLE OF INHIBITING BIOSYNTHESIS OF PARASITE'S ANCHORING GROUP WASHINGTON UNIVERSITY (US) 1998-06-02 US disclosed
US-5747537-A Method of inhibiting parasitic activity WASHINGTON UNIVERSITY (US) 1998-05-05 US disclosed