Sunitinib

Sunitinib

SCHEMBL8082

CCN(CC)CCNC(=O)c1c(C)[nH]c(C=C2C(=O)Nc3ccc(F)cc32)c1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CSF1RFLT1FLT3FLT4KDRKITPDGFRAPDGFRBRET

The experimentally established mechanism targets of Sunitinib. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR known ✓ P35968 16/20 1.00
PDGFRB known ✓ P09619 7/20 1.00
CSF1R known ✓ P07333 3/20 1.00
FLT3 known ✓ P36888 3/20 1.00
RET known ✓ P07949 2/20 1.00
FLT4 known ✓ P35916 2/20 1.00
KIT known ✓ P10721 2/20 1.00
PDGFRA known ✓ P16234 1/20 1.00
FLT1 known ✓ P17948 1/20 1.00
PRKAA1 Q13131 13/20 1.00
PRKAA2 P54646 12/20 1.00
FGFR1 P11362 5/20 1.00
EGFR P00533 3/20 1.00
PLK4 O00444 2/20 1.00
DCLK1 O15075 2/20 1.00
PDPK1 O15530 2/20 1.00
DAPK3 O43293 2/20 1.00
ROCK2 O75116 2/20 1.00
RPS6KA5 O75582 2/20 1.00
RPS6KA4 O75676 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sunitinib SCHEMBL25343935 1.00 KDR (1.00) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL20805212 1.00 KDR (1.00) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL30314241 1.00 KDR (1.00) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL25343938 1.00 KDR (1.00) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL8081 1.00 KDR (1.00) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL2296353 0.99 KDR (0.98) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL23668540 0.99 KDR (0.98) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL28454734 0.99 KDR (0.98) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL2716609 0.99 KDR (0.98) KDRPRKAA1PRKAA2PDGFRBFGFR1
Sunitinib SCHEMBL1780287 0.98 KDR (0.97) KDRPRKAA1PRKAA2PDGFRBFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 73959 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144750-A1 Dosing Regimens for Treatment of Glioblastoma SIGNPATH PHARMA INC. (US) 2026-05-28 US claimed
US-20260144866-A1 METHODS, DEVICES, AND SYSTEMS FOR PREDICTING TREATMENT RESPONSIVENESS OF CLEAR CELL RENAL CELL CARCINOMA PATIENTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-05-28 US claimed
EP-3836899-B1 CHEMOTHERAPEUTIC PHARMACEUTICAL SUSPENSION FOR ORAL DOSAGE ONCOSOL LTD (GB) 2026-05-27 EP claimed
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
CN-116162546-B Drug screening tumor organoid chip and drug screening method DALIAN INSTITUTE OF CHEMICAL PHYSICS, CHINESE ACADEMY OF SCIENCES (CN) 2026-05-26 CN claimed
CN-122075716-A Medicine for treating tumor by combining recombinant oncolytic virus and small-molecule anticancer medicine 2026-05-26 CN claimed
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
CN-122075735-A Therapeutic combinations comprising anti-FOLR 1 immunoconjugates 2026-05-26 CN claimed
CN-122074048-A Methods of treating cancer 诺华股份有限公司 2026-05-22 CN claimed
WO-2026105121-A1 ANTICANCER FORMULATIONS AND USES THEREOF INTRAGEL THERAPEUTICS LTD. (IL) 2026-05-21 WO claimed
WO-2006084869-A1 TETRAHYDROPYRIDOTHIOPHENES FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER NYCOMED GMBH (DE) 2006-08-17 WO claimed
WO-2006079645-A1 NOVEL INDOLOPYRIDINES , BENZOFURANOPYRIDINES AND BENZOTHIENOPYRIDINES NYCOMED GMBH (DE) 2006-08-03 WO claimed
WO-2006079644-A1 INDOLOPYRIDINES, BENZOFURANOPYRIDINES AND BENZOTHIENOPYRIDINES NYCOMED GMBH (DE) 2006-08-03 WO claimed
WO-2006075012-A2 PYRROLODIHYDROISOQUINOLINES AS ANTIPROLIFERATIVE AGENTS NYCOMED GMBH (DE) 2006-07-20 WO claimed
WO-2006027346-A2 NOVEL PYRAZOLOPYRIMIDINES ALTANA PHARMA AG (DE) 2006-03-16 WO claimed
JP-2005503386-A 2005-02-03 JP claimed
US-20040152759-A1 Combination administration of an indolinone with a chemotherapeutic agent for cell proliferation disorders SUGEN, INC. 2004-08-05 US claimed
EP-1419151-A1 CHRYSTALS INCLUDING A MALIC ACID SALT OF N-[2-(DIETHYLAMINO)ETHYL]-5-[(5-FLUORO-1,2-DIHYDRO-2-OXO-3H-INDOLE-3-YLIDENE)METHYL]-2,4-DIMETHYL-1H-PYRROLE-3-CARBOXAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS THEREOF PHARMACIA & UPJOHN COMPANY (US) 2004-05-19 EP claimed
US-20030069298-A1 Crystals including a malic acid salt of a 3-pyrrole substituted 2-indolinone, and compositions thereof PHARMACIA & UPJOHN COMPANY 2003-04-10 US claimed
WO-2003016305-A1 CRYSTALS INCLUDING A MALIC ACID SALT OF N-[2-(DIETHYLAMINO) ETHYL]-5-[(5-FLUORO-2-OXO-3H-INDOLE-3-YLIDENE) METHYL]-2, 4-DIMETHYL-1H-PYRROLE-3-CARBOXAMIDE, PROCESSES FOR ITS PREPARATION AND COMPOSITIONS THEREOF PHARMACIA & UPJOHN COMPANY (US) 2003-02-27 WO claimed