SCHEMBL8083452

SCHEMBL8083452

CCc1ccc(CNC(=O)c2cc(-c3cc(C)cc(F)c3)cnc2-c2cccnn2)cc1OC

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 18/20 0.67
HCRTR1 O43613 16/20 0.67
HTR1A P08908 1/20 0.49
OPRM1 P35372 1/20 0.49
DRD3 P35462 1/20 0.49
HTR2B P41595 1/20 0.49
KCNH2 Q12809 1/20 0.49
LMNA P02545 1/20 0.42
CYP3A4 P08684 1/20 0.40
HTR2A P28223 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12024836 0.93 HCRTR2 (0.77) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL3487028 0.80 HCRTR2 (0.60) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL3622483 0.80 HCRTR2 (1.00) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL3023755 0.78 HCRTR2 (0.62) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL8086304 0.76 HCRTR2 (0.72) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL8081046 0.75 HCRTR2 (0.73) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL13498698 0.75 HCRTR2 (0.69) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL13499116 0.75 HCRTR2 (0.56) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL3622904 0.75 HCRTR1 (1.00) HCRTR2HCRTR1HTR1AOPRM1DRD3
SCHEMBL14548868 0.74 HCRTR2 (0.56) HCRTR2HCRTR1HTR1AOPRM1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020642-A1 PYRIDINE CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2009-02-12 WO disclosed