SCHEMBL8084466

SCHEMBL8084466

C[C@]12CCC(=O)NC1CC[C@@H]1[C@H]2CC[C@]2(C)C(c3ccccc3)CC[C@@H]12

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 5/20 0.63
SRD5A1 P18405 3/20 0.63
AR P10275 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084464 1.00 SRD5A2 (0.63) SRD5A2SRD5A1AR
SCHEMBL8710566 0.90 SRD5A1 (0.55) SRD5A2SRD5A1AR
SCHEMBL8023123 0.87 SRD5A1 (0.53) SRD5A2SRD5A1AR
SCHEMBL8020698 0.87 SRD5A1 (0.53) SRD5A2SRD5A1AR
SCHEMBL8006582 0.86 SRD5A1 (0.52) SRD5A2SRD5A1AR
SCHEMBL8019047 0.85 SRD5A2 (0.51) SRD5A2SRD5A1AR
SCHEMBL8019119 0.84 SRD5A2 (0.56) SRD5A2SRD5A1AR
SCHEMBL8650910 0.84 SRD5A2 (0.53) SRD5A2SRD5A1AR
SCHEMBL8650908 0.84 SRD5A2 (0.53) SRD5A2SRD5A1AR
SCHEMBL8023090 0.83 SRD5A2 (0.55) SRD5A2SRD5A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0756481-B1 17$g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO INC (US) 2000-12-27 EP disclosed
EP-0756481-A4 17-g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO INC (US) 1998-11-18 EP disclosed
EP-0756481-A1 17$g(b)-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO. INC. (US) 1997-02-05 EP disclosed
US-5525608-A ANTIACNE AGENT, SKIN DISORDERS, GLANDULAR DISORDERS MERCK & CO., INC. (US) 1996-06-11 US disclosed
WO-1995028928-A1 17β-ARYL-4-AZA-STEROID DERIVATIVES MERCK & CO., INC. (US) 1995-11-02 WO disclosed