SCHEMBL8086085

SCHEMBL8086085

NC(C(=O)N(CCc1ccc(C(F)(F)F)cc1)c1ccc(O)cc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.42
GLI1 P08151 2/20 0.40
GLI2 P10070 2/20 0.40
MLYCD O95822 5/20 0.39
SLC6A9 P48067 1/20 0.39
PDPK1 O15530 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
PDK2 Q15119 1/20 0.37
PDK4 Q16654 1/20 0.37
PLAAT3 P53816 1/20 0.37
PLAAT5 Q96KN8 1/20 0.37
PLAAT2 Q9NWW9 1/20 0.37
PLAAT4 Q9UL19 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3649918 0.90 TACR1 (0.44) TACR1MLYCDSLC6A9PDPK1MEN1
SCHEMBL3645573 0.90 PTGIR (0.43) TACR1MLYCDSLC6A9PDPK1MEN1
SCHEMBL3645993 0.90 TACR1 (0.44) TACR1MLYCDSLC6A9PDPK1MEN1
SCHEMBL3645996 0.90 TACR1 (0.44) TACR1MLYCDSLC6A9PDPK1MEN1
SCHEMBL8082608 0.88 TACR1 (0.43) TACR1GLI1GLI2SLC6A9PDPK1
SCHEMBL4155415 0.87 SERPINE1 (0.44) TACR1SLC6A9
SCHEMBL3642140 0.87 CHRM5 (0.45) TACR1SLC6A9MEN1KMT2A
SCHEMBL3644592 0.86 PPARG (0.45) TACR1SLC6A9
SCHEMBL3649784 0.86 PPARG (0.45) TACR1SLC6A9
SCHEMBL3644589 0.86 PPARG (0.45) TACR1SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016087-A1 MONOAMIDE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 WO disclosed