SCHEMBL8086189

SCHEMBL8086189

O=C1N(C[C@H](O)COc2ccc(NS(=O)O)cc2)CCN1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.51
GRIN2B Q13224 2/20 0.51
MAPT P10636 5/20 0.43
HTT P42858 1/20 0.43
KCNH2 Q12809 7/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
CACNA1G O43497 3/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ATF4 P18848 3/20 0.37
RECQL P46063 1/20 0.37
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009654 0.85 GRIN1 (0.49) GRIN1GRIN2BMAPTHTTKCNH2
SCHEMBL12576447 0.84 GRIN1 (0.51) GRIN1GRIN2BMAPTHTTKCNH2
SCHEMBL2016246 0.84 GRIN1 (0.72) GRIN1GRIN2BKCNH2
SCHEMBL2016248 0.84 GRIN1 (0.72) GRIN1GRIN2BKCNH2
SCHEMBL14864160 0.75 GRIN1 (0.54) GRIN1GRIN2BMAPTHTTKCNH2
SCHEMBL12576482 0.74 MAPT (0.68) MAPTHTTKCNH2LMNASMN1; SMN2
SCHEMBL2023658 0.74 KCNH2 (0.68) MAPTHTTKCNH2CACNA1GLMNA
SCHEMBL2023657 0.74 KCNH2 (0.68) MAPTHTTKCNH2CACNA1GLMNA
SCHEMBL2025770 0.74 KCNH2 (0.61) MAPTKCNH2DRD2DRD3CACNA1G
SCHEMBL2025768 0.74 KCNH2 (0.61) MAPTKCNH2DRD2DRD3CACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006437-A1 NMDA RECEPTOR ANTAGONISTS FOR NEUROPROTECTION EMORY UNIVERSITY (US) 2009-01-08 WO disclosed