SCHEMBL8091007

SCHEMBL8091007

NCC1CC=CC2CN(c3nc4c(cc3F)c(=O)c(C(=O)O)cn4C3CC3)CC21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.58
CHRM2 P08172 2/20 0.58
DRD1 P21728 1/20 0.58
LMNA P02545 3/20 0.54
KDM4E B2RXH2 2/20 0.54
HSD17B10 Q99714 2/20 0.54
ABCC4 O15439 1/20 0.54
EPHA2 P29317 1/20 0.48
FLT4 P35916 1/20 0.48
GSK3B P49841 1/20 0.48
RARB P10826 1/20 0.48
TBXAS1 P24557 1/20 0.48
SLC6A3 Q01959 1/20 0.48
DHFR P00374 1/20 0.46
ALDH1A1 P00352 2/20 0.45
POLB P06746 2/20 0.45
HPGD P15428 1/20 0.45
XBP1 P17861 1/20 0.45
NFKB1 P19838 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9046917 0.90 DPP4 (0.48) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL8083243 0.89 DPP4 (0.65) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL8091078 0.85 DPP4 (0.56) DPP4CHRM2DRD1LMNAKDM4E
Trovafloxacin9 SCHEMBL9186378 0.85 DPP4 (0.66) DPP4CHRM2DRD1LMNAKDM4E
Trovafloxacin9 SCHEMBL9186361 0.85 DPP4 (0.66) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL8083142 0.85 DPP4 (0.49) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL10668511 0.84 DPP4 (0.64) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL10668501 0.84 DPP4 (0.64) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL10511561 0.84 DPP4 (0.64) DPP4CHRM2DRD1LMNAKDM4E
SCHEMBL8094753 0.83 KDM4E (0.57) LMNAKDM4EHSD17B10ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018054-A INTERMEDIATE COMPOUNDS FOR PREPARING NOVEL QUINOLONE AND NAPHTHYRIDONE DERIVATIVES WHICH ARE SUBSTITUTED IN THE 7-POSITION BY A PARTIALLY HYDROGENATED ISOINDOLINYL RING, USE AS ANTIBACTERIAL AGENTS AND AS FEED ADDITIVES BAYER AKTIENGESELLSCHAFT (DE) 2000-01-25 US disclosed