SCHEMBL8091121

SCHEMBL8091121

O=[N+]([O-])c1cnc2ccc(SCCNCc3ccnc(CSc4nc5ccccc5[nH]4)c3Cl)nn12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.38
NPC1 O15118 5/20 0.38
RAB9A P51151 5/20 0.38
LMNA P02545 3/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
HTT P42858 1/20 0.37
CYP1A2 P05177 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2E1 P05181 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP3A4 P08684 1/20 0.34
HPGD P15428 5/20 0.33
ALDH1A1 P00352 3/20 0.33
PSMD14 O00487 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8503009 0.85
SCHEMBL8091117 0.83 MAPT (0.32) LMNAMAPTHTTALDH1A1MEN1
SCHEMBL8091119 0.83 MAPT (0.38) SMN1; SMN2NPC1RAB9ALMNAMAPT
Hydrochloric Acid SCHEMBL8092772 0.79 NPC1 (0.42) SMN1; SMN2NPC1RAB9ALMNAMAPT
Hydrochloric Acid SCHEMBL8089347 0.74 MAPT (0.37) SMN1; SMN2NPC1RAB9ALMNAMAPT
SCHEMBL9232763 0.73 MAPT (0.49) SMN1; SMN2NPC1RAB9ALMNAMAPT
Hydrochloric Acid SCHEMBL8089324 0.73 MAPT (0.37) SMN1; SMN2NPC1RAB9ALMNAMAPT
SCHEMBL8089354 0.69 MEN1 (0.34) SMN1; SMN2NPC1RAB9ALMNAMAPT
Hydrochloric Acid SCHEMBL8089345 0.69 MKNK1 (0.30)
Hydrochloric Acid SCHEMBL8092773 0.69 MAPT (0.32) SMN1; SMN2NPC1RAB9ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043242-A TREATING A MAMMAL AFFLICTED WITH A DISEASE BASED ON HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2000-03-28 US disclosed
EP-0946559-A2 IMIDAZOPYRIDAZINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1999-10-06 EP disclosed
WO-1998028299-A2 IMIDAZOPYRIDAZINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1998-07-02 WO disclosed