SCHEMBL8091326

SCHEMBL8091326

CS(=O)(=O)Nc1ccc(S(N)(=O)=O)cc1OC1CCCCC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.67
PTGS2 P35354 3/20 0.67
ALDH1A1 P00352 2/20 0.67
PTGS1 P23219 2/20 0.67
MEN1 O00255 1/20 0.67
PTGES O14684 1/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2D6 P10635 1/20 0.67
MAPT P10636 1/20 0.67
ALOX15 P16050 1/20 0.67
TSHR P16473 1/20 0.67
CYP2C19 P33261 1/20 0.67
KMT2A Q03164 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
YAP1 P46937 1/20 0.49
S1PR1 P21453 1/20 0.47
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ns-398 SCHEMBL9505682 0.81 CYP19A1 (0.98) CYP19A1PTGS2ALDH1A1PTGS1MEN1
Ns-398 SCHEMBL214213 0.80 CYP19A1 (1.00) CYP19A1PTGS2ALDH1A1PTGS1MEN1
SCHEMBL9504767 0.80 CYP19A1 (1.00) CYP19A1PTGS2ALDH1A1PTGS1MEN1
Ns-398 SCHEMBL29368077 0.80 CYP19A1 (1.00) CYP19A1PTGS2ALDH1A1PTGS1MEN1
Ns-398 SCHEMBL9505633 0.79 CYP19A1 (0.98) CYP19A1PTGS2ALDH1A1PTGS1MEN1
Ns-398 SCHEMBL9505672 0.79 CYP19A1 (0.98) CYP19A1PTGS2ALDH1A1PTGS1MEN1
Ns-398 SCHEMBL9505669 0.79 CYP19A1 (0.98) CYP19A1PTGS2ALDH1A1PTGS1MEN1
Ns-398 SCHEMBL9505627 0.79 CYP19A1 (0.98) CYP19A1PTGS2ALDH1A1PTGS1MEN1
SCHEMBL3296493 0.79 CYP19A1 (1.00) CYP19A1PTGS2ALDH1A1PTGS1MEN1
SCHEMBL8523784 0.78 PTGS1 (0.61) CYP19A1PTGS2ALDH1A1PTGS1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed
EP-0848703-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II Nycomed Austria GmbH (AT) 1998-06-24 EP disclosed
WO-1997003953-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 1997-02-06 WO disclosed