SCHEMBL8092301

SCHEMBL8092301

CCc1cc(C2O[C@@H](n3cnc4c(NCCC5CCCCC5)nc(N[C@H](CO)Cc5ccccc5)nc43)[C@H](OC=O)[C@@H]2O)on1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.47
ADORA3 P0DMS8 4/20 0.42
ADORA1 P30542 3/20 0.42
ADORA2B P29275 1/20 0.42
CDK1 P06493 3/20 0.40
CDK5 Q00535 2/20 0.40
PGK1 P00558 1/20 0.39
PGK2 P07205 1/20 0.39
CCNE1 P24864 2/20 0.39
CDK2 P24941 2/20 0.39
CCNE2 O96020 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6943628 1.00 ADORA2A (0.47) ADORA2AADORA3ADORA1ADORA2BCDK1
SCHEMBL6839820 0.91 ADORA2A (0.53) ADORA2AADORA3ADORA1ADORA2BCDK1
SCHEMBL6839786 0.89 ADORA2A (0.46) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7104786 0.87 ADORA2A (0.47) ADORA2AADORA3ADORA1ADORA2BCDK1
SCHEMBL7595823 0.84 ADORA1 (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL6839047 0.82 ADORA2A (0.45) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL6841752 0.80 ADORA2A (0.51) ADORA2AADORA3ADORA1ADORA2BCDK1
SCHEMBL6839112 0.79 ADORA2A (0.50) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7104998 0.79 ADORA2A (0.47) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL7601339 0.79 ADORA2A (0.56) ADORA2AADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051425-A2 2-(PURIN-9-yl)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-11-15 EP disclosed
WO-1999038877-A2 2-(PURIN-9-yl)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES GLAXO GROUP LIMITED (GB) 1999-08-05 WO disclosed