SCHEMBL8092362

SCHEMBL8092362

C[C@H]1COCCN1c1cc(CS(C)(=O)=O)nc(-c2ccc3c(N)c[nH]c3c2)n1

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.71
MTOR P42345 10/20 0.71
PIK3CD O00329 4/20 0.64
ATR Q13535 9/20 0.55
CYP2C9 P11712 1/20 0.52
PDCD1 Q15116 6/20 0.49
CD274 Q9NZQ7 6/20 0.49
ATRIP Q8WXE1 5/20 0.49
CHEK1 O14757 4/20 0.49
PDPK1 O15530 2/20 0.49
ROCK1 Q13464 2/20 0.49
AURKB Q96GD4 2/20 0.49
AURKA O14965 1/20 0.49
PRKDC P78527 1/20 0.47
ATM Q13315 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3081794 0.89 PIK3CA (0.66) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL3082179 0.88 PIK3CA (0.70) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL3082131 0.86 PIK3CA (0.88) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL3076902 0.84 PIK3CA (0.69) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL3093063 0.84 PIK3CA (0.71) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL3600666 0.84 PIK3CA (0.70) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL739897 0.83 PIK3CA (0.72) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL3095615 0.83 PIK3CA (1.00) PIK3CAMTORPIK3CDATRCYP2C9
SCHEMBL3601400 0.83 PIK3CA (0.67) PIK3CAMTORPIK3CDATRPDCD1
SCHEMBL3083758 0.83 PIK3CA (1.00) PIK3CAMTORPIK3CDATRCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007751-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed