SCHEMBL8092640

SCHEMBL8092640

COC(=O)C(OC)(c1ccccc1)C(C)c1ccc(SC)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.43
KIF11 P52732 1/20 0.40
ALDH1A1 P00352 2/20 0.37
EDNRB P24530 2/20 0.37
EDNRA P25101 2/20 0.37
AKR1C3 P42330 3/20 0.37
AKR1C2 P52895 3/20 0.37
ACACB O00763 1/20 0.36
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
SRC P12931 1/20 0.34
CES1 P23141 1/20 0.34
NPC1 O15118 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28626535 0.76 KCNN4 (0.49) KCNN4ALDH1A1MEN1KMT2ALMNA
SCHEMBL618735 0.73 KMT2A (0.44) KCNN4KMT2ALMNAKDM4ESMN1; SMN2
SCHEMBL28261002 0.67 HPGD (0.49) ALDH1A1AKR1C3AKR1C2ACACBKMT2A
SCHEMBL10717798 0.67 CYP1A2 (0.52) KCNN4KIF11ALDH1A1EDNRBEDNRA
SCHEMBL1470523 0.66 CES1 (0.73) KCNN4KIF11ALDH1A1EDNRBEDNRA
SCHEMBL1626673 0.66 PLK1 (0.47) KCNN4KIF11ALDH1A1LMNASMN1; SMN2
SCHEMBL16713397 0.64 CYP2D6 (0.49) KCNN4KIF11KMT2ALMNAKDM4E
SCHEMBL3931951 0.64 KCNN4 (0.67) KCNN4ALDH1A1MEN1KMT2AOPRM1
SCHEMBL27564046 0.64 KCNN4 (0.60) KCNN4KIF11MEN1KMT2AOPRM1
SCHEMBL18095170 0.63 SRC (0.46) KCNN4ALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882015-B1 DIPHENYL STILBENES AS PRODRUGS TO COX-2 INHIBITORS MERCK FROSST CANADA INC (CA) 2000-12-27 EP disclosed
EP-0882015-A1 DIPHENYL STILBENES AS PRODRUGS TO COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1998-12-09 EP disclosed
US-5733909-A ANTIINFLAMMATORY AGENTS; ANALGESICS; ANTIPYRETIC AGENT MERCK FROSST CANADA, INC. (CA) 1998-03-31 US disclosed
WO-1997028120-A1 DIPHENYL STILBENES AS PRODRUGS TO COX-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1997-08-07 WO disclosed