SCHEMBL8093323

SCHEMBL8093323

CNS(=O)(=O)Cc1ccc2[nH]cc(CCN3CC[C@@H](CNCc4ccccc4)C3)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 20/20 1.00
HTR1B P28222 20/20 1.00
HTR1A P08908 5/20 1.00
HTR2A P28223 5/20 1.00
HTR2C P28335 1/20 0.50
HTR1E P28566 1/20 0.50
HTR1F P30939 1/20 0.50
HTR7 P34969 1/20 0.50
HTR2B P41595 1/20 0.50
HTR3A P46098 1/20 0.50
HTR5A P47898 1/20 0.50
SLC47A1 Q96FL8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7474847 0.90 HTR1D (0.82) HTR1DHTR1BHTR1AHTR2A
SCHEMBL7478803 0.81 HTR1D (1.00) HTR1DHTR1BHTR1AHTR2A
SCHEMBL7478800 0.81 HTR1D (1.00) HTR1DHTR1BHTR1AHTR2A
Methylamine SCHEMBL8096304 0.80 HTR1D (0.66) HTR1DHTR1BHTR1AHTR2A
SCHEMBL7481032 0.79 HTR1D (0.66) HTR1DHTR1BHTR1AHTR2A
SCHEMBL4578602 0.79 HTR1D (1.00) HTR1DHTR1BHTR1AHTR2AHTR2C
SCHEMBL4358113 0.79 HTR1D (1.00) HTR1DHTR1BHTR1AHTR2A
SCHEMBL4578911 0.79 HTR1D (1.00) HTR1DHTR1BHTR1AHTR2A
SCHEMBL4358107 0.79 HTR1D (1.00) HTR1DHTR1BHTR1AHTR2A
SCHEMBL9047260 0.77 HTR1D (0.66) HTR1DHTR1BHTR1AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6025374-A Azetidine, pyrrolidine and piperidine derivatives as 5HT1 receptor agonists MERCK SHARP & DOHME, LTD. (GB) 2000-02-15 US disclosed