SCHEMBL8093574

SCHEMBL8093574

CCCCCCCCCCNCCCCCCCCCC.CN[C@H](C)c1ccccc1.N#CCCNCc1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.52
SCN8A Q9UQD0 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8728583 0.88 CHRM2 (0.68) CHRM2SCN8AL3MBTL1ALDH1A1NPSR1
SCHEMBL10556589 0.77 CHRM2 (0.81) CHRM2SCN8AL3MBTL1ALDH1A1NPSR1
SCHEMBL19509215 0.77 CHRM2 (0.81) CHRM2SCN8AL3MBTL1ALDH1A1NPSR1
SCHEMBL11083068 0.77 CHRM2 (0.81) CHRM2SCN8AL3MBTL1ALDH1A1NPSR1
SCHEMBL728747 0.76 CYP1A2 (0.65) CHRM2SCN8AALDH1A1NPSR1CYP1A2
SCHEMBL2188249 0.76 CHRM2 (0.78) CHRM2SCN8AL3MBTL1ALDH1A1NPSR1
SCHEMBL2711100 0.72 CHRM2 (0.75) CHRM2SCN8AL3MBTL1ALDH1A1NPSR1
SCHEMBL27299308 0.72 CYP1A2 (0.54) CHRM2L3MBTL1ALDH1A1NPSR1CYP1A2
SCHEMBL11594897 0.69 CHRM2 (0.93) CHRM2SCN8AALDH1A1NPSR1CYP1A2
SCHEMBL27298367 0.69 CHRM2 (0.69) CHRM2SCN8AL3MBTL1ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed