SCHEMBL8095567

SCHEMBL8095567

Nc1cc(C2(S(=O)(=O)C3CCOCC3)CC2)nc(-c2ccc(NC(=O)NC3CCC3)cc2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 5/20 0.45
MTOR P42345 3/20 0.45
PIK3CA P42336 3/20 0.45
PIK3CB P42338 1/20 0.45
PIK3CG P48736 1/20 0.45
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
RAB9A P51151 3/20 0.40
GAA P10253 2/20 0.40
EPHX1 P07099 2/20 0.40
NPC1 O15118 2/20 0.39
KIT P10721 1/20 0.38
KDR P35968 1/20 0.38
FLT3 P36888 1/20 0.38
ATR Q13535 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RICTOR Q6R327 1/20 0.37
MAPKAP1 Q9BPZ7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092188 0.92 PIK3CA (0.45) PIK3CDMTORPIK3CAPIK3CBPIK3CG
SCHEMBL8096200 0.92 EPHX1 (0.47) CA12CA1CA2CA9RAB9A
SCHEMBL8091090 0.91 PIK3CD (0.45) PIK3CDMTORPIK3CAPIK3CBPIK3CG
SCHEMBL8084603 0.90 PIK3CA (0.46) PIK3CDMTORPIK3CAPIK3CBPIK3CG
SCHEMBL8081909 0.90 CA12 (0.41) PIK3CDMTORPIK3CAPIK3CBPIK3CG
SCHEMBL8091695 0.90 CA12 (0.41) PIK3CDMTORPIK3CAPIK3CBPIK3CG
SCHEMBL8092629 0.89 MTOR (0.48) PIK3CDMTORPIK3CAPIK3CBPIK3CG
SCHEMBL8098257 0.87 PIK3CD (0.48) PIK3CDMTORPIK3CAPIK3CBPIK3CG
SCHEMBL8099411 0.86 CA12 (0.44) PIK3CDCA12CA1CA2CA9
SCHEMBL4203492 0.85 PIK3CA (0.54) PIK3CDMTORPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed