SCHEMBL8097346

SCHEMBL8097346

N#Cc1ccc(Cc2cnc(Cc3ccc(-c4ccccc4F)cc3)[nH]2)cc1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 16/20 0.61
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
HRH3 Q9Y5N1 1/20 0.41
PDE10A Q9Y233 1/20 0.38
DAO P14920 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104996 0.87 BRS3 (0.62) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7927590 0.86 BRS3 (0.61) BRS3HRH3PDE10A
Hydrochloric Acid SCHEMBL8307429 0.86 BRS3 (0.61) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7921316 0.86 BRS3 (0.61) BRS3CYP11B1CYP11B2HRH3
SCHEMBL7919370 0.85 BRS3 (0.58) BRS3HRH3PDE10A
SCHEMBL7919393 0.85 BRS3 (0.62) BRS3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8310488 0.84 BRS3 (0.57) BRS3HRH3PDE10A
SCHEMBL8305740 0.84 BRS3 (0.59) BRS3CYP11B1CYP11B2HRH3
SCHEMBL8107240 0.84 BRS3 (0.62) BRS3PDE10A
SCHEMBL8110784 0.84 BRS3 (0.59) BRS3HRH3PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP claimed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO claimed