SCHEMBL8098541

SCHEMBL8098541

COc1ccc(F)c(C2CC2)c1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 9/20 0.46
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
DPP4 P27487 2/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
IDH2 P48735 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21644922 0.92 FFAR1 (0.45) FFAR1HTR2AHTR2CHTR2BPTGDR2
SCHEMBL20103281 0.91 PTGDR2 (0.52) FFAR1HTR2AHTR2CHTR2BPTGDR2
SCHEMBL21644868 0.87 FFAR1 (0.51) FFAR1PTGDR2SLC6A4
SCHEMBL21644953 0.87 FFAR1 (0.45) FFAR1PTGDR2DPP4
SCHEMBL20103540 0.87 FFAR1 (0.51) FFAR1PTGDR2SLC6A4
SCHEMBL24645999 0.87 FFAR1 (0.47) FFAR1HTR2APTGDR2SLC6A4
SCHEMBL20103513 0.87 FFAR1 (0.51) FFAR1PTGDR2SLC6A4
SCHEMBL20103493 0.87 FFAR1 (0.45) FFAR1PTGDR2DPP4
SCHEMBL20103517 0.87 FFAR1 (0.51) FFAR1PTGDR2SLC6A4
SCHEMBL20103359 0.87 FFAR1 (0.45) FFAR1PTGDR2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105492429-A Heteroaryl inhibitors of SUMO activating enzyme MILLENNIUM PHARM INC 2016-04-13 CN disclosed
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed