SCHEMBL8099622

SCHEMBL8099622

COc1cc(N2CCN[C@H](C)C2)ccc1C

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KHK P50053 2/20 0.47
TLR9 Q9NR96 1/20 0.46
TLR8 Q9NR97 1/20 0.46
TLR7 Q9NYK1 1/20 0.46
CHEK1 O14757 1/20 0.46
GHSR Q92847 2/20 0.45
MAPT P10636 2/20 0.45
DPP4 P27487 3/20 0.44
ADRB1 P08588 1/20 0.43
TGFBR1 P36897 1/20 0.41
ACVR1 Q04771 1/20 0.41
BCL2A1 Q16548 2/20 0.40
BRPF1 P55201 2/20 0.40
BRD4 O60885 1/20 0.40
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2243476 0.88 TLR9 (0.55) KHKTLR9TLR8TLR7CHEK1
SCHEMBL8270689 0.88 TLR9 (0.55) KHKTLR9TLR8TLR7CHEK1
Hydrochloric Acid SCHEMBL4572995 0.87 TLR9 (0.54) KHKTLR9TLR8TLR7CHEK1
SCHEMBL2867159 0.84 BCL2A1 (0.50) KHKTLR9TLR8TLR7CHEK1
SCHEMBL13066645 0.84 TLR9 (0.47) KHKTLR9TLR8TLR7CHEK1
SCHEMBL1639654 0.84 BCL2A1 (0.50) KHKTLR9TLR8TLR7CHEK1
SCHEMBL2873748 0.84 CHEK1 (0.47) KHKTLR9TLR8TLR7CHEK1
SCHEMBL1639658 0.84 BCL2A1 (0.50) KHKTLR9TLR8TLR7CHEK1
SCHEMBL2873745 0.84 CHEK1 (0.47) KHKTLR9TLR8TLR7CHEK1
SCHEMBL8110949 0.84 TLR9 (0.45) KHKTLR9TLR8TLR7CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001127-A1 CYANOCYCLOPROPYLCARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed