SCHEMBL810219

SCHEMBL810219

N#CNC(=NCCCCCCCCCCOc1cccc(Cl)c1)Nc1cccnc1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 9/20 0.62
CYP3A4 P08684 2/20 0.62
CYP2D6 P10635 2/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
NOTUM Q6P988 2/20 0.55
EGFR P00533 6/20 0.51
ABCC9 O60706 4/20 0.47
ABCC8 Q09428 4/20 0.47
KCNJ11 Q14654 4/20 0.47
KCNJ8 Q15842 4/20 0.47
P2RX7 Q99572 1/20 0.46
MEN1 O00255 1/20 0.45
CYP1A2 P05177 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPK1 P28482 2/20 0.44
TSHR P16473 1/20 0.44
QPCT Q16769 1/20 0.43
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL810331 1.00 NAMPT (0.62) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL810207 1.00 NAMPT (0.62) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL810083 1.00 NAMPT (0.62) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL810074 1.00 NAMPT (0.62) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL809999 0.89 NAMPT (0.78) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL810038 0.89 NAMPT (0.78) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL810341 0.89 NAMPT (0.78) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL810190 0.89 NAMPT (0.78) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL811109 0.89 NAMPT (0.78) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL810352 0.89 NAMPT (0.78) NAMPTCYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394649-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDYL CYANOGUANIDINES, PREPARATION METHODS AND USES THEREOF Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2011-12-14 EP claimed
EP-2394649-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING PYRIDYL CYANOGUANIDINES, PREPARATION METHODS AND USES THEREOF Tianjin Hemay Bio-Tech Co., Ltd. (CN) 2011-12-14 EP disclosed