SCHEMBL8102964

SCHEMBL8102964

CC(C)N(CCOc1ccc2cc(C(=O)O)ccc2c1)C(C)C

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.53
ESR2 Q92731 2/20 0.53
MCHR1 Q99705 3/20 0.53
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 1/20 0.50
THRA P10827 1/20 0.49
LTA4H P09960 1/20 0.49
MAPK1 P28482 1/20 0.49
RARB P10826 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2741668 0.87 ESR1 (0.64) ESR1ESR2MCHR1LTA4HMAPK1
SCHEMBL8176484 0.86 MAPT (0.51) ESR1ESR2MCHR1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL224473 0.85 ESR1 (0.62) ESR1ESR2MCHR1LTA4HMAPK1
SCHEMBL8134642 0.84 KDM4E (0.69) ESR1KDM4EALDH1A1THRA
SCHEMBL465181 0.82 KDM4E (0.65) KDM4ETHRARARB
SCHEMBL30726463 0.82 KDM4E (0.65) KDM4ETHRARARB
SCHEMBL465148 0.82 KDM4E (0.65) KDM4ETHRAMAPK1RARB
SCHEMBL8092814 0.82 BCHE (0.56) ESR1KDM4EALDH1A1THRA
SCHEMBL8189320 0.80 MCHR1 (0.49) ESR1ESR2MCHR1THRA
SCHEMBL8084842 0.80 KDM4E (0.62) KDM4ETHRARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810206-B1 Substituted 2-naphthoylguanidines, process for their preparation, their use as medicament or diagnostic agent and medicament containing them HOECHST AG (DE) 2000-12-27 EP disclosed
US-6087304-A ANTIARRHYTHMIC PHARMACEUTICALS HAVING A CARDIOPROTECTIVE COMPONENT FOR INFARCT PROPHYLAXIS AND INFARCT TREATMENT AND FOR THE TREATMENT OF ANGINA PECTORIS HOECHST AKTIENGESELLSCHAFT (DE) 2000-07-11 US disclosed
EP-0810206-A1 Substituted 2-naphtoylguanidines, process for their preparation, their use as medicament or diagnostic agent and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-12-03 EP disclosed