SCHEMBL8105364

SCHEMBL8105364

O=S(=O)(Nc1cncc(-c2ccc3nccc(-c4ccncc4)c3c2)c1)C1C=NNC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 15/20 0.57
AKT1 P31749 3/20 0.57
MTOR P42345 4/20 0.44
PIK3CD O00329 3/20 0.44
PIK3CB P42338 3/20 0.44
PIK3CG P48736 3/20 0.44
PIK3C3 Q8NEB9 2/20 0.44
MAPK10 P53779 1/20 0.42
CLK2 P49760 2/20 0.37
DYRK1A Q13627 2/20 0.37
CLK3 P49761 1/20 0.37
GAK O14976 1/20 0.36
RPS6KA4 O75676 1/20 0.36
STK10 O94804 1/20 0.36
PIM1 P11309 1/20 0.36
CSNK2A2 P19784 1/20 0.36
MAP2K2 P36507 1/20 0.36
CSNK1D P48730 1/20 0.36
CLK1 P49759 1/20 0.36
CSNK1G2 P78368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL729588 0.84 PIK3CA (0.64) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL8119215 0.78 PIK3CA (0.57) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL14024679 0.78 PIK3CA (0.57) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL729945 0.78 PIK3CA (0.66) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL731497 0.77 PIK3CA (0.65) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL8132469 0.77 PIK3CA (0.53) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL729752 0.76 PIK3CA (0.62) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL8121050 0.76 PIK3CA (0.55) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL731678 0.76 PIK3CA (0.75) PIK3CAAKT1MTORPIK3CDPIK3CB
SCHEMBL741238 0.75 PIK3CA (0.74) PIK3CAAKT1MTORPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008144463-A1 QUINOLINE DERIVATIVES AS PI3 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-11-27 WO disclosed