SCHEMBL8105902

SCHEMBL8105902

COc1ccc(Br)cc1COCC1(c2ccccc2)CCNCC1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 17/20 0.60
SLC6A4 P31645 6/20 0.56
KCNH2 Q12809 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1388687 0.99 TACR1 (0.58) TACR1SLC6A4KCNH2
SCHEMBL3595110 0.82 TACR1 (0.48) TACR1SLC6A4KCNH2
SCHEMBL3596809 0.82 TACR1 (0.54) TACR1SLC6A4KCNH2
SCHEMBL3589377 0.81 TACR1 (0.59) TACR1
SCHEMBL8124474 0.79 TACR1 (0.59) TACR1SLC6A4KCNH2
Hydrochloric Acid SCHEMBL1388317 0.78 TACR1 (0.58) TACR1SLC6A4KCNH2
SCHEMBL3590159 0.78 TACR1 (0.60) TACR1SLC6A4KCNH2
SCHEMBL3596983 0.77 TACR1 (0.49) TACR1SLC6A4KCNH2
SCHEMBL5446697 0.77 TACR1 (0.49) TACR1SLC6A4KCNH2
SCHEMBL14403909 0.77 TACR1 (0.49) TACR1SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0666856-B1 4-ARYLMETHYLOXYMETHYL PIPERIDINES AS TACHYKININ ANTAGONISTS MERCK SHARP & DOHME (GB) 2000-01-05 EP claimed