SCHEMBL8106771

SCHEMBL8106771

C[C@@H](n1ncn(-c2ccc(OCC(F)(F)C(F)F)cc2)c1=O)[C@@](O)(C=O)c1ccc(F)cc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 14/20 0.37
CYP2C9 P11712 11/20 0.37
CYP2C19 P33261 10/20 0.37
CYP1A2 P05177 6/20 0.37
CYP2D6 P10635 6/20 0.37
ABCB11 O95342 1/20 0.36
CYP17A1 P05093 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
PTGS2 P35354 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
CYP8B1 Q9UNU6 1/20 0.36
MAPT P10636 1/20 0.34
UGCG Q16739 1/20 0.34
KCNH2 Q12809 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PPARD Q03181 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106768 1.00 CYP3A4 (0.37) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8097530 0.88 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8097526 0.88 CYP3A4 (0.38) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL19970517 0.84 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL1456168 0.84 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL19970516 0.84 CYP3A4 (0.51) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8111174 0.84 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8107346 0.84 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8107262 0.83 CYP3A4 (0.37) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL8107260 0.83 CYP3A4 (0.37) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1033367-A2 Process for the preparation of optically active triazole derivatives and their imidazolidin-2-one intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-06 EP disclosed
US-5677464-A Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0687672-A2 Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-20 EP disclosed