SCHEMBL8107071

SCHEMBL8107071

N#Cc1ccc(Cc2cnc(Cc3ccc(-c4ccccc4)c(N)n3)[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 11/20 0.54
AOC3 Q16853 1/20 0.40
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
GHSR Q92847 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8303919 0.99 BRS3 (0.53) BRS3AOC3CYP11B1CYP11B2HRH3
SCHEMBL8303912 0.88 BRS3 (0.55) BRS3AOC3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8303557 0.88 BRS3 (0.54) BRS3AOC3CYP11B1CYP11B2HRH3
SCHEMBL8308371 0.81 BRS3 (0.56) BRS3AOC3CYP11B1CYP11B2HRH3
SCHEMBL7919393 0.81 BRS3 (0.62) BRS3AOC3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8304730 0.81 BRS3 (0.55) BRS3AOC3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8521500 0.80 BRS3 (0.61) BRS3AOC3CYP11B1CYP11B2HRH3
SCHEMBL8307560 0.79 BRS3 (0.54) BRS3AOC3CYP11B1CYP11B2HRH3
SCHEMBL7919373 0.79 BRS3 (0.56) BRS3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8522033 0.78 BRS3 (0.53) BRS3AOC3CYP11B1CYP11B2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP claimed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO claimed
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP disclosed
EP-0891361-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO disclosed
WO-1997036901-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed