SCHEMBL8109484

SCHEMBL8109484

CCOC(=O)CN(C(=O)c1ccccn1)c1ccc2c(c1)nc(CNc1ccc(C#N)cc1)n2C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.53
F2 P00734 10/20 0.46
NR1I2 O75469 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
SLC6A2 P23975 1/20 0.46
AGTR1 P30556 1/20 0.46
SLC6A3 Q01959 1/20 0.46
SCN5A Q14524 1/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SLC22A2 O15244 1/20 0.44
F10 P00742 1/20 0.44
PLG P00747 1/20 0.44
PLAT P00750 1/20 0.44
PROC P04070 1/20 0.44
HPN P05981 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
PRSS3 P35030 1/20 0.44
SLC47A2 Q86VL8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6636532 0.89 F2 (0.53) NQO2F2NR1I2ADORA3SLC6A2
SCHEMBL6636973 0.88 NQO2 (0.69) NQO2F2NR1I2ADORA3SLC6A2
SCHEMBL6775703 0.85 NQO2 (0.70) NQO2F2NR1I2ADORA3SLC6A2
SCHEMBL6781191 0.85 F2 (0.64) NQO2F2NR1I2ADORA3SLC6A2
SCHEMBL28719520 0.82 NQO2 (0.62) NQO2F2NR1I2ADORA3SLC6A2
SCHEMBL6635444 0.82 F2 (0.48) NQO2F2NPC1RAB9AHDAC6
SCHEMBL505917 0.80 NQO2 (0.82) NQO2F2NR1I2ADORA3SLC6A2
Hydrochloric Acid SCHEMBL14696865 0.79 NQO2 (0.81) NQO2F2NR1I2ADORA3SLC6A2
SCHEMBL6780051 0.78 F2 (0.63) NQO2F2NR1I2ADORA3SLC6A2
Oxalic Acid SCHEMBL13684738 0.78 NQO2 (0.79) NQO2F2NR1I2ADORA3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6121308-A INDOLE AND BENZIMIDAZOLE ANTITHROMBOTIC COMPOUNDS, SUCH AS 1-METHYL-2-(N-(4-AMIDINOPHENYL)-AMINOMETHYL)-5-(N-(HYDROXYCARBONYLMETHYL) -QUINOLINE-8-SULPHONYLAMINO)-INDOLE BOEHRINGER INGELHEIM KG (DE) 2000-09-19 US disclosed