SCHEMBL8116170

SCHEMBL8116170

CCCc1cc(C(=O)OC)ccc1OC(C(=O)NS(=O)(=O)c1cccc2cccnc12)c1ccc2c(c1)OCO2

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 14/20 0.59
EDNRB P24530 12/20 0.59
AGTR1 P30556 3/20 0.48
LMNA P02545 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
GAA P10253 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ITGB3 P05106 1/20 0.44
ITGAV P06756 1/20 0.44
ALDH1A1 P00352 2/20 0.44
AGTR2 P50052 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7332607 0.94 EDNRA (0.68) EDNRAEDNRBAGTR1LMNATP53
SCHEMBL7335601 0.88 EDNRA (0.52) EDNRAEDNRBAGTR1LMNACYP1A2
SCHEMBL5494850 0.87 EDNRA (0.65) EDNRAEDNRBAGTR1SMN1; SMN2ALDH1A1
SCHEMBL5496424 0.86 EDNRA (0.65) EDNRAEDNRBAGTR1AGTR2
SCHEMBL5489155 0.85 EDNRA (0.66) EDNRAEDNRBAGTR1GAAAGTR2
SCHEMBL7330600 0.84 EDNRA (0.77) EDNRAEDNRBAGTR1AGTR2
SCHEMBL7335276 0.82 EDNRA (0.73) EDNRAEDNRBAGTR1
SCHEMBL7339608 0.82 EDNRA (0.69) EDNRAEDNRBAGTR1TSHRSMN1; SMN2
SCHEMBL7329183 0.81 EDNRA (0.86) EDNRAEDNRBAGTR1AGTR2
SCHEMBL7333529 0.81 EDNRA (0.76) EDNRAEDNRBAGTR1SMN1; SMN2AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0617001-B1 Phenoxyphenylacetic acid derivatives MERCK & CO INC (US) 2000-01-26 EP claimed