SCHEMBL8123239

SCHEMBL8123239

COC(=O)c1ccc(O)c(Br)c1.COC(=O)c1ccc(OC(C)C)c(Br)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.51
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
CA7 P43166 3/20 0.51
CA9 Q16790 3/20 0.51
CA14 Q9ULX7 3/20 0.51
XDH P47989 1/20 0.51
NOTUM Q6P988 1/20 0.50
ESR1 P03372 1/20 0.47
ALDH1A1 P00352 5/20 0.47
MAPT P10636 3/20 0.47
ALOX12 P18054 2/20 0.47
KDM4E B2RXH2 2/20 0.47
HSD17B10 Q99714 2/20 0.47
HPGD P15428 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.47
ALOX15 P16050 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1980076 0.93 NOTUM (0.56) CA12CA1CA2CA7CA9
SCHEMBL29550817 0.85 CA1 (0.69) CA12CA1CA2CA7CA9
SCHEMBL382159 0.85 CA1 (0.69) CA12CA1CA2CA7CA9
SCHEMBL978911 0.81 NOTUM (0.53) CA12CA1CA2CA7CA9
SCHEMBL403444 0.81 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL21437595 0.80 NOTUM (0.49) CA12CA1CA2CA7CA9
SCHEMBL31063212 0.80 NOTUM (0.55) CA12CA1CA2CA7CA9
SCHEMBL8163137 0.80 NOTUM (0.55) CA12CA1CA2CA7CA9
SCHEMBL10088910 0.78 NOTUM (0.57) CA12CA1CA2CA7CA9
SCHEMBL401131 0.77 KMT2A (0.53) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986559-A1 1,6-NAPHTHYRIDINE ANTI-CONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-03-22 EP disclosed
WO-1998054184-A1 1,6-NAPHTHYRIDINE ANTI-CONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1998-12-03 WO disclosed