SCHEMBL8130561

SCHEMBL8130561

CCN(CC)CCNc1ncc2cc(-c3c(Cl)cccc3Cl)c(N)nc2n1

nearest known ligand 0.89

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 20/20 0.89
KDR P35968 1/20 0.60
EGFR P00533 5/20 0.59
SRC P12931 5/20 0.59
FGFR2 P21802 4/20 0.59
FGFR4 P22455 4/20 0.59
FGFR3 P22607 4/20 0.59
PRKD3 O94806 1/20 0.57
PRKCG P05129 1/20 0.57
PRKCB P05771 1/20 0.57
PRKCA P17252 1/20 0.57
PRKCH P24723 1/20 0.57
PRKCI P41743 1/20 0.57
PRKCE Q02156 1/20 0.57
PRKCQ Q04759 1/20 0.57
PRKCZ Q05513 1/20 0.57
PRKCD Q05655 1/20 0.57
PRKD1 Q15139 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8122918 0.94 FGFR1 (1.00) FGFR1KDREGFRSRCFGFR2
SCHEMBL8131809 0.93 FGFR1 (0.94) FGFR1KDREGFRSRCFGFR2
SCHEMBL8127223 0.88 FGFR1 (0.89) FGFR1KDREGFRSRCFGFR2
SCHEMBL8804236 0.87 FGFR1 (0.91) FGFR1KDREGFRSRCFGFR2
SCHEMBL8131641 0.85 FGFR1 (0.81) FGFR1KDREGFRSRCFGFR2
SCHEMBL8138254 0.83 FGFR1 (1.00) FGFR1KDREGFRSRCFGFR2
SCHEMBL8804686 0.82 FGFR1 (0.91) FGFR1KDREGFRSRCFGFR2
SCHEMBL8130391 0.82 FGFR1 (1.00) FGFR1KDREGFRSRCFGFR2
SCHEMBL140148 0.80 FGFR1 (1.00) FGFR1KDREGFRSRCFGFR2
SCHEMBL144578 0.79 FGFR1 (1.00) FGFR1KDREGFRSRCFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790997-B1 6-ARYL PYRIDO[2,3-d]PYRIMIDINES AND NAPHTHYRIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2000-03-22 EP disclosed
EP-0790997-A2 6-ARYL PYRIDO( 2,3-d]PYRIMIDINES AND NAPHTHYRIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1997-08-27 EP disclosed
WO-1996015128-A2 6-ARYL PYRIDO[2,3-d]PYRIMIDINES AND NAPHTHYRIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-05-23 WO disclosed