SCHEMBL8134702

SCHEMBL8134702

CC(=O)Oc1cc(OCc2ccc3c(c2)OCO3)ccc1C#N

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
CYP3A4 P08684 1/20 0.52
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8807149 0.90 NPC1 (0.48) NPC1RAB9ACYP3A4KMT2AMEN1
SCHEMBL8807664 0.86 AR (0.47) NPC1RAB9ACYP3A4
SCHEMBL8133441 0.83 NPC1 (0.54) NPC1RAB9ACYP3A4MAOB
SCHEMBL8807681 0.82 NPC1 (0.53) NPC1RAB9AMAOB
SCHEMBL8124618 0.80
SCHEMBL8807145 0.79 NPC1 (0.44) NPC1RAB9AMAOB
SCHEMBL8133504 0.79 NPC1 (0.53) NPC1RAB9AMAOB
SCHEMBL8809410 0.79 MRGPRX4 (0.49) MAOB
SCHEMBL8117951 0.79
SCHEMBL8117947 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124343-A Substituted phenyl compounds with a substituent having a thienyl ring RHONE-POULENC RORER LIMITED (GB) 2000-09-26 US disclosed
EP-0805802-B1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LTD (GB) 2000-08-16 EP disclosed
US-6048893-A Substituted phenyl compounds with a substituent having A 1,3-benzodioxole ring RHONE-POULENC RORER LIMITED (GB) 2000-04-11 US disclosed
EP-0805802-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE-POULENC RORER LIMITED (GB) 1997-11-12 EP disclosed
WO-1996022978-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LIMITED (GB) 1996-08-01 WO disclosed