SCHEMBL8136171

SCHEMBL8136171

B.OC(c1ccccc1)(c1ccccc1)[C@@H]1CCCN1

nearest known ligand 0.93

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.93
MAPK1 P28482 2/20 0.93
KDM4E B2RXH2 1/20 0.93
NPC1 O15118 1/20 0.93
CYP1A2 P05177 1/20 0.93
HPGD P15428 1/20 0.93
CYP2C19 P33261 1/20 0.93
RAB9A P51151 1/20 0.93
LMNA P02545 3/20 0.51
MEN1 O00255 1/20 0.51
HRH1 P35367 1/20 0.51
SCN1A P35498 1/20 0.51
KMT2A Q03164 1/20 0.51
SCN2A Q99250 1/20 0.51
SCN3A Q9NY46 1/20 0.51
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CHRM3 P20309 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL100361 0.98 CYP2D6 (0.96) CYP2D6MAPK1KDM4ENPC1CYP1A2
SCHEMBL239738 0.98 CYP2D6 (0.96) CYP2D6MAPK1KDM4ENPC1CYP1A2
SCHEMBL100360 0.98 CYP2D6 (0.96) CYP2D6MAPK1KDM4ENPC1CYP1A2
SCHEMBL7446968 0.96 CYP2D6 (0.93) CYP2D6MAPK1KDM4ENPC1CYP1A2
Hydrochloric Acid SCHEMBL9277459 0.96 CYP2D6 (1.00) CYP2D6MAPK1KDM4ENPC1CYP1A2
Pipradrol SCHEMBL156360 0.93 CYP2D6 (0.87) CYP2D6MAPK1KDM4ENPC1CYP1A2
Pipradrol SCHEMBL4057811 0.91 CYP2D6 (0.90) CYP2D6MAPK1KDM4ENPC1CYP1A2
Sulfuric Acid SCHEMBL9452303 0.90 CYP2D6 (0.82) CYP2D6MAPK1KDM4ENPC1CYP1A2
SCHEMBL6295242 0.89 CYP2D6 (0.79) CYP2D6MAPK1KDM4ENPC1CYP1A2
SCHEMBL5054811 0.89 CYP2D6 (0.79) CYP2D6MAPK1KDM4ENPC1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668266-B1 Process for preparing 1,1-diarylprolinols MERCK & CO INC (US) 2000-02-02 EP disclosed
EP-0962451-A2 Chiral catalysts for reduction of ketones and process for their preparation MERCK & CO. INC. (US) 1999-12-08 EP disclosed
EP-0668266-A1 Chiral catalysts for reduction of ketones and process for their preparation MERCK & CO. INC. (US) 1995-08-23 EP disclosed
US-5264585-A Reaction of diarylmethanol with boroxanine MERCK & CO., INC. (US) 1993-11-23 US disclosed
US-5189177-A Chiral boron catalysts for reduction of ketones and process for their preparation MERCK & CO., INC. (US) 1993-02-23 US disclosed
EP-0453298-A2 Chiral catalysts for reduction of ketones and process for their preparation MERCK & CO. INC. (US) 1991-10-23 EP disclosed
US-5039802-A Arylation process for preparation of chiral catalysts for ketone reduction MERCK & CO., INC. (US) 1991-08-13 US disclosed